反应条件
1: 6-bromo-1,3-dihydro-2H-indol-2-one With n-butyllithium; N,N,N',N,-tetramethylethylenediamine in tetrahydrofuran 2: 1,5-diiodo-3-oxa-pentane in tetrahydrofuran T=-78 - 20°C;
参考文献
Eastwood, Paul; Gonzalez, Jacob; Gomez, Elena; Caturla, Francisco; Balague, Cristina; Orellana, Adelina; Dominguez, Maria
Bioorganic and Medicinal Chemistry Letters, 2011 , vol. 21, # 18 p. 5270 - 5273