2-氨基-3-甲基-5-溴吡啶合成路线

参考文献

Watterson, Scott H.; Chen, Ping; Zhao, Yufen; Gu, Henry H.; Dhar, T. G. Murali; Xiao, Zili; Ballentine, Shelley K.; Shen, Zhongqi; Fleener, Catherine A.; Rouleau, Katherine A.; Obermeier, Mary; Yang, Zheng; McIntyre, Kim W.; Shuster, David J.; Witmer, Mark; Dambach, Donna; Chao, Sam; Mathur, Arvind; Chen, Bang-Chi; Barrish, Joel C.; Robl, Jeffrey A.; Townsend, Robert; Iwanowicz, Edwin J.
Journal of Medicinal Chemistry, 2007 , vol. 50, # 15 p. 3730 - 3742

3430-21-52-氨基-3-甲基-5-溴吡啶

1033439-60-9

参考文献

Tremblay, Martin; Bonneau, Pierre; Bousquet, Yves; Deroy, Patrick; Duan, Jianmin; Duplessis, Martin; Gagnon, Alexandre; Garneau, Michel; Goudreau, Nathalie; Guse, Ingrid; Hucke, Oliver; Kawai, Stephen H.; Lemke, Christopher T.; Mason, Stephen W.; Simoneau, Bruno; Surprenant, Simon; Titolo, Steve; Yoakim, Christiane
Bioorganic and Medicinal Chemistry Letters, 2012 , vol. 22, # 24 p. 7512 - 7517

3430-21-52-氨基-3-甲基-5-溴吡啶

142404-81-72-乙酰氨基-5-溴-3-甲基吡啶

参考文献

PFIZER INC.
Patent: EP842924 A1, 1998 ;
EP 0842924 A1

3430-21-52-氨基-3-甲基-5-溴吡啶+

75-36-5乙酰氯

142404-81-72-乙酰氨基-5-溴-3-甲基吡啶

参考文献

Fujisawa Pharmaceutical Co., Ltd.
Patent: US6083961 A1, 2000 ;

3430-21-52-氨基-3-甲基-5-溴吡啶+

73183-34-3联硼酸频那醇酯

1111637-91-23-甲基-5-(4,4,5,5-四甲基-1,3,2-二噁硼烷-2-基)吡啶-2-胺

参考文献

IRM LLC; NOVARTIS AG; CHATTERJEE, Arnab Kumar; NAGLE, Advait Suresh; PARASELLI, Prasuna; KONDREDDI, Ravinder Reddy; LEONG, Seh Yong; MISHRA, Pranab Kumar; MOREAU, Robert Joseph; ROLAND, Jason Thomas; SIM, Wei Lin Sandra; SIMON, Oliver; TAN, Liying Jocelyn; YEUNG, Bryan KS; ZOU, Bin; BOLLU, Venkatataiah
Patent: WO2014/78802 A1, 2014 ;
Location in patent: Page/Page column 71; 94; 95 ;

3430-21-52-氨基-3-甲基-5-溴吡啶

166266-19-92-氨基-3-甲基-5-碘吡啶

参考文献

US2006/69093 A1, ;

Page/Page column 23 ;
US 20060069093 A1

3430-21-52-氨基-3-甲基-5-溴吡啶

167626-78-06-氨基-5-甲基烟酸

参考文献

WO2013/42139 A1, ;

3430-21-52-氨基-3-甲基-5-溴吡啶

156072-86-55-溴-3-甲基-2-吡啶甲腈

参考文献

CUSHMAN, Mark S.; KISELEV, Evgeny A.; MORRELL, Andrew E.
Patent: US2014/18360 A1, 2014 ;

557-21-1氰化锌+

3430-21-52-氨基-3-甲基-5-溴吡啶

183428-91-3

参考文献

ADVINUS THERAPEUTICS LIMITED; KHARUL, Rajendra; BHUNIYA, Debnath; MOOKHTIAR, Kasim A.; SINGH, Umesh; HAZARE, Atul; PATIL, Satish; DATRANGE, Laxmikant; THAKKAR, Mahesh
Patent: WO2013/42139 A1, 2013 ;
Location in patent: Page/Page column 83 ;

544-92-3氰化亚铜+

3430-21-52-氨基-3-甲基-5-溴吡啶

183428-91-3

参考文献

Boykin, David W.; Tidwell, Richard R.; Wilson, W. David; Ismail, Mohamed A.
Patent: US2005/282853 A1, 2005 ;
Location in patent: Page/Page column 20 ;