1: With 4-methylmorpholine N-oxide in toluene; acetonitrile T=-10°C; 0.5 - 1 h; 2: With ammonia; water in toluene; acetonitrile Product distribution / selectivity;
参考文献
ASTRAZENECA AB
Patent: WO2008/136745 A1, 2008 ;
Location in patent: Page/Page column 14-15 ;