1: Cs2CO3 / dimethylformamide / 1.5 h 2: Et3N / CH2Cl2 / -78 - 20 °C View Scheme
参考文献
Anderson, Marc O.; Sherrill, John; Madrid, Peter B.; Liou, Ally P.; Weisman, Jennifer L.; DeRisi, Joseph L.; Guy, R. Kiplin
Bioorganic and Medicinal Chemistry, 2006 , vol. 14, # 2 p. 334 - 343