反应条件
1: 85 percent / 2,4-bis(4-methoxyphenyl)-2,4-dithioxo-1,3,2,4-dithiadiphosphetane / hexamethylphosphoric acid triamide / 6 h / 100 °C
2: 90 percent / SnCl2*2H2O / ethanol / 4 h / Heating
3: 70 percent / ICl, AcOH / 1.5 h / 25 °C
View Scheme
参考文献
Shi, Dong-Fang; Bradshaw, Tracey D.; Wrigley, Samantha; McCall, Carol J.; Lelieveld, Peter; Fichtner, Iduna; Stevens, Malcolm F. G.
Journal of Medicinal Chemistry, 1996 , vol. 39, # 17 p. 3375 - 3384