反应条件
4-(N,N-dimethlyamino)pyridine; triethylamine in N,N-dimethyl-formamide T=0 - 20°C; 1 h; regioselective reaction;
参考文献
Herdemann, Matthias; Weber, Alexander; Jonveaux, Jerome; Schwoebel, Frank; Stoeck, Michael; Heit, Isabelle
Bioorganic and Medicinal Chemistry Letters, 2011 , vol. 21, # 6 p. 1852 - 1856