2-氟苯胺合成路线

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Saavedra, Oscar; Claridge, Stephen; Zhan, Lijie; Raeppel, Franck; Granger, Marie-Claude; Raeppel, Stephane; Mannion, Michael; Gaudette, Frederic; Zhou, Nancy; Isakovic, Ljubomir; Bernstein, Naomy; Deziel, Robert; Nguyen, Hannah; Beaulieu, Normand; Beaulieu, Carole; Dupont, Isabelle; Wang, James; Macleod, A. Robert; Besterman, Jeffrey M.; Vaisburg, Arkadii
Bioorganic and Medicinal Chemistry Letters, 2009 , vol. 19, # 24 p. 6836 - 6839

348-54-92-氟苯胺+

61436-88-22-溴-N-甲基苯甲酰胺

92152-36-8

参考文献

Baars, Hannah; Beyer, Astrid; Kohlhepp, Stefanie V.; Bolm, Carsten
Organic Letters, 2014 , vol. 16, # 2 p. 536 - 539

348-54-92-氟苯胺+

73365-02-3BOC-D-脯氨醛

924907-26-6(R)-1-boc-2-[(2-氟苯基氨基)-甲基]-吡咯烷

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MERCK PATENT GMBH
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348-54-92-氟苯胺

93129-68-1N-(4-氰基-2-氟苯基)乙酰胺

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Kruger; Keck; Noll; Pieper
Arzneimittel-Forschung/Drug Research, 1984 , vol. 34, # 11 A p. 1612 - 1624

348-54-92-氟苯胺

97760-94-6N-(2-氟-4-碘苯基)乙酰氨

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Kruger; Keck; Noll; Pieper
Arzneimittel-Forschung/Drug Research, 1984 , vol. 34, # 11 A p. 1612 - 1624

348-54-92-氟苯胺+

123-73-9巴豆醛

46001-36-98-氟-2-甲基喹啉

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GLAXO GROUP LIMITED; GORE, Paul Martin; HANCOCK, Ashley, Paul; HODGSON, Simon Teanby
Patent: WO2010/94643 A1, 2010 ;
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WO 2010/094643 A1

123-73-9巴豆醛+

348-54-92-氟苯胺

46001-36-98-氟-2-甲基喹啉

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Clavier, Sylvain; Rist, ystein; Hansen, Stina; Gerlach, Lars-Ole; Hoegberg, Thomas; Bergman, Jan
Organic and Biomolecular Chemistry, 2003 , vol. 1, # 23 p. 4248 - 4253

66023-21-0+

348-54-92-氟苯胺

46001-36-98-氟-2-甲基喹啉

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Recordati S.A.
Patent: US2003/162777 A1, 2003 ;
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348-54-92-氟苯胺

46001-36-98-氟-2-甲基喹啉

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Chandrashekarappa, Kiran Kumar H.; Mahadevan, Kittappa M.; Manjappa, Kiran B.
Tetrahedron Letters, 2013 , vol. 54, # 11 p. 1368 - 1370

38520-78-4+

348-54-92-氟苯胺

49579-08-0

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Welch; Ewing; Huang; Menniti; Pagnozzi; Kelly; Seymour; Guanowsky; Guhan; Guinn; Critchett; Lazzaro; Ganong; DeVries; Staigers; Chenard
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