反应条件
1: 4.5 g / Pd(OAc)2, Ph3P, KOAc, nBu4NCl / dimethylformamide / 24 h / 80 °C 2: 4.1 g / H2 / 10percent Pd/C / ethanol / 3 h / 2585.7 Torr / Ambient temperature View Scheme
参考文献
Rosenblum, Stuart B.; Huynh, Tram; Afonso, Adriano; Davis Jr., Harry R.; Yumibe, Nathan; Clader, John W.; Burnett, Duane A.
Journal of Medicinal Chemistry, 1998 , vol. 41, # 6 p. 973 - 980