1-(5-硝基吡啶-2-基)哌啶-4-醇合成路线 （共 6 条）
反应条件
in propan-1-ol T=100°C; 1.5 h;
参考文献
Daiichi Asubio Pharma Co., Ltd.
Patent: EP1775298 A1, 2007 ;
Location in patent: Page/Page column 35 ;
反应条件
N-ethyl-N,N-diisopropylamine in N,N-dimethyl-formamide T=100°C;
参考文献
Ting, Pauline C.; Lee, Joe F.; Zorn, Nicolas; Kim, Hyunjin M.; Aslanian, Robert G.; Lin, Mingxiang; Smith, Michelle; Walker, Scott S.; Cook, John; Van Heek, Margaret; Lachowicz, Jean
Bioorganic and Medicinal Chemistry Letters, 2013 , vol. 23, # 4 p. 985 - 988
参考文献
US2011/224137 A1, ;
US 20110224137 A1
反应条件
1: N-ethyl-N,N-diisopropylamine / ethanol View Scheme
参考文献
US2011/224137 A1, ;
US 20110224137 A1
反应条件
1: N-ethyl-N,N-diisopropylamine / ethanol View Scheme
参考文献
US2011/224137 A1, ;
US 20110224137 A1
反应条件
hydrogen; palladium 10 on activated carbon in ethanol
T=20°C; 3 h;
参考文献
BRISTOL-MYERS SQUIBB COMPANY; DEVASTHALE, Pratik; WASHBURN, William N.; RENDUCHINTALA, Kishore V.; SRIDHAR, Radhakrishnan
Patent: WO2010/42682 A1, 2010 ;
Location in patent: Page/Page column 71 ;
WO 2010/042682 A1
