反应条件
hydrogenchloride; sodium hydroxide; 1-ethyl-(3-(3-dimethylamino)propyl)-carbodiimide hydrochloride 1.) dioxane, H2O, RT, 4 h, 2.) dioxane, H2O, reflux, 10 min; Yield given. Multistep reaction;
参考文献
Journal of medicinal chemistry, , vol. 35, # 16 p. 3066 - 3075