反应条件
1: 57.7 percent / m-chloroperbenzoic acid, p-TsOH*H2O / CH2Cl2 / 3 h / Ambient temperature 2: 1.) K2CO3, 2.) tetra-n-butylammonium iodide / 1.) DMF, 2.) DMF, RT 3: 11.5 mg / H2 / 10percent Pd-C / tetrahydrofuran / 2792.6 Torr View Scheme
参考文献
Journal of Medicinal Chemistry, , vol. 38, # 12 p. 2041 - 2049