1: With diisobutylaluminium hydride in tetrahydrofuran; toluene T=-78°C; 2.16667 h; 2: With hydrogenchloride; ethanol; water in tetrahydrofuran; toluene 3: With sodium tetrahydroborate; water; sodium hydrogencarbonate more than 3 stages;
参考文献
Pfizer Inc
Patent: US2007/270438 A1, 2007 ;
Location in patent: Page/Page column 35 ;
US 20070270438 A1