Piotrowski, David W.; Rogers, Bruce N.; McWhorter JR., William W.; Walker, Daniel Patrick; Corbett, Jeffrey W.; Groppi JR., Vincent E.; Rudmann, Daniel G.
Patent: US2003/236287 A1, 2003 ;
Location in patent: Page 44 ;
US 20030236287 A1
1: 42 percent / toluene / 4.5 h / 100 - 110 °C
2: 77 percent / POCl3 / 0.5 h / Heating
3: 69 percent / pyridine hydrochloride / 2-ethoxy-ethanol / 3 h / 120 °C
View Scheme
参考文献
Boschelli, Diane H.; Wang, Yanong D.; Johnson, Steve; Wu, Biqi; Ye, Fei; Barrios Sosa, Ana Carolina; Golas, Jennifer M.; Boschelli, Frank
Journal of Medicinal Chemistry, 2004 , vol. 47, # 7 p. 1599 - 1601