5-(4-甲氧基苯基)-3-苯基-1,2-恶唑合成路线 (共 43 条)
反应条件
lead(IV) acetate in benzene
4 h; Heating;
参考文献
Sharma, T. C.; Rojindar, S.; Berge, D. D.; Kale, A. V.
Indian Journal of Chemistry, Section B: Organic Chemistry Including Medicinal Chemistry, 1986 , vol. 25, p. 437
反应条件
sulfuric acid in acetic acid
Heating;
参考文献
Day, Ruth Ann; Blake, Jacqueline A.; Stephens, Chad E.
Synthesis, 2003 , # 10 p. 1586 - 1590
反应条件
methanol; hydroxylamine hydrochloride
参考文献
Weygand; Bauer
Justus Liebigs Annalen der Chemie, 1927 , vol. 459, p. 143
反应条件
chloroform; tris-(2-chloro-ethyl)-amine
参考文献
Tuerck; Behringer
Chemische Berichte, 1965 , vol. 98, p. 3020,3023
反应条件
hydroxylamine hydrochloride in methanol
24 h; Heating; Yield given. Yields of byproduct given. Title compound not separated from byproducts;
参考文献
Bandiera, T.; Gruenanger, P.; Albini, F. Marinone
Journal of Heterocyclic Chemistry, 1992 , vol. 29, # 6 p. 1423 - 1428
反应条件
in various solvent(s)
Heating;
参考文献
Baranski, Andrzej; Cholewka, Elzbieta
Polish Journal of Chemistry, 1989 , vol. 63, # 4-12 p. 483 - 494
反应条件
sulfuric acid in acetic acid
Heating;
参考文献
Day, Ruth Ann; Blake, Jacqueline A.; Stephens, Chad E.
Synthesis, 2003 , # 10 p. 1586 - 1590
反应条件
1: N-chlorosuccinimide / dimethylformamide / 0 °C
2: triethylamine / ethyl acetate
View Scheme
参考文献
Weidner-Wells, Michele A.; Henninger, Todd C.; Fraga-Spano, Stephanie A.; Boggs, Christine M.; Matheis, Michele; Ritchie, David M.; Argentieri, Dennis C.; Wachter, Michael P.; Hlasta, Dennis J.
Bioorganic and Medicinal Chemistry Letters, 2004 , vol. 14, # 16 p. 4307 - 4311
反应条件
triethylamine in ethyl acetate
参考文献
Weidner-Wells, Michele A.; Henninger, Todd C.; Fraga-Spano, Stephanie A.; Boggs, Christine M.; Matheis, Michele; Ritchie, David M.; Argentieri, Dennis C.; Wachter, Michael P.; Hlasta, Dennis J.
Bioorganic and Medicinal Chemistry Letters, 2004 , vol. 14, # 16 p. 4307 - 4311
反应条件
1: 95 percent / TFA / 4 h / 20 °C
2: 73 percent / γ-MnO2 / benzene / 2 h / Heating
View Scheme
参考文献
Saginova, L. G.; Kukhareva, I. L.; Lebedev, A. T.; Shabarov, Yu. S.
Journal of Organic Chemistry USSR (English Translation), 1991 , vol. 27, # 9.1 p. 1631 - 1638
Zhurnal Organicheskoi Khimii, 1991 , vol. 27, # 9 p. 1852 - 1860