4-氯吡咯并嘧啶合成路线

346599-63-14-氯-5,7-二氢-6H-吡咯并[2,3-D]嘧啶-6-酮

参考文献

Sun; Cui, Jean; Liang, Congxin; Zhou, Yong; Nematalla, Asaad; Wang, Xueyan; Chen, Hui; Tang, Cho; Wei, James
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3680-69-14-氯吡咯并嘧啶

60129-59-1（2R，3S，5R）-5-（4-氨基-7H-吡咯[2,3-D]嘧啶-7-基-2 -（羟甲基）四氢呋喃-3-醇

参考文献

Kazimierczuk, Zygmunt; Cottam, Howard B.; Revankar, Ganapathi R.; Robins, Roland K.
Journal of the American Chemical Society, 1984 , vol. 106, # 21 p. 6379 - 6382

3680-69-14-氯吡咯并嘧啶

941685-27-44-(1H-吡唑-4-基)-7-((2-(三甲基甲硅烷基)乙氧基)-甲基)-7h-吡咯并[2,3-d]嘧啶

参考文献

INCYTE CORPORATION; ZHOU, Jiacheng; LIU, Pingli; CAO, Ganfeng; WU, Yongzhong
Patent: WO2013/36611 A1, 2013 ;

76513-69-42-(三甲基硅烷基)乙氧甲基氯+

3680-69-14-氯吡咯并嘧啶

941685-26-34-CHLORO-7-((2-(TRIMETHYLSILYL)ETHOXY)METHYL)-7H-PYRROLO[2,3-D]PYRIMIDINE

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Zhou, Jiacheng; Liu, Pingli; Lin, Qiyan; Metcalf, Brian W.; Meloni, David; Pan, Yongchun; Xia, Michael; Li, Mei; Yue, Tai-Yuen; Rodgers, James D.; Wang, Haisheng
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1146629-84-6(βR)-β-环戊基-4-(4,4,5,5-四甲基-1,3,2-二氧杂硼杂环戊烷-2-基)-1H-吡唑-1-丙腈+

3680-69-14-氯吡咯并嘧啶

941678-49-5鲁索替尼

参考文献

Zhou, Jiacheng; Liu, Pingli; Lin, Qiyan; Metcalf, Brian W.; Meloni, David; Pan, Yongchun; Xia, Michael; Li, Mei; Yue, Tai-Yuen; Rodgers, James D.; Wang, Haisheng
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3680-69-14-氯吡咯并嘧啶+

98-59-9对甲苯磺酰氯

479633-63-14-氯-7-甲苯磺酰基-7H-吡咯[2,3-D]嘧啶

参考文献

WO2010/123919 A2, ;

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137-43-9溴代环戊烷+

3680-69-14-氯吡咯并嘧啶

212268-44-54-氯-7-环戊基-7H-吡咯并[2,3-d]嘧啶

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PFIZER PRODUCTS INC.
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3680-69-14-氯吡咯并嘧啶

212268-44-54-氯-7-环戊基-7H-吡咯并[2,3-d]嘧啶

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Sobolov, Susan B.; Sun, Jianmin; Cooper, Beth A.
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98-09-9苯磺酰氯+

3680-69-14-氯吡咯并嘧啶

186519-89-14-氯-7-(苯基磺酰基)-7h-吡咯并[2,3-d]嘧啶

参考文献

Mayasundari, Anand; Fujii, Naoaki
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3680-69-14-氯吡咯并嘧啶

252723-17-47-苯磺酰基-5-溴-4-氯-7H-吡咯并[2,3-d]嘧啶

参考文献

CONVERGENCE PHARMACEUTICALS LIMITED; WITTY, David R.; NORTON, David; TIERNEY, Jason Paul; LORTHIOIR, Ghislaine; SIME, Mairi; PHILPOTT, Karen Louise
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