ammonium hydroxide in water
T=140°C; 2 h; Microwave irradiationInert atmosphere; Overall yield = 57 percent; Overall yield = 378 mg;
参考文献
Verheij, Mark H. P.; Thompson, Andrew J.; Van Muijlwijk-Koezen, Jacqueline E.; Lummis, Sarah C. R.; Leurs, Rob; De Esch, Iwan J. P.
Journal of Medicinal Chemistry, 2012 , vol. 55, # 20 p. 8603 - 8614