反应条件
1: COCl2 / tetrahydrofuran / 18 h / Ambient temperature 2: 60.5 percent / CHCl3; tetrahydrofuran / a) RT, 2 h, b) reflux, 2 h View Scheme
参考文献
Perricone; Humphrey; Skaletzky; Graham; Zandt; Zins
Journal of Medicinal Chemistry, 1994 , vol. 37, # 22 p. 3693 - 3700