反应条件
1: 1.) sodium methoxide / 1.) methanol, 0 deg C, 2.) DMF, 25 deg C
2: iron, glacial acetic acid / methanol / 5.5 h / Heating
View Scheme
参考文献
Duncia, John V.; Chiu, Andrew T.; Carini, David J.; Gregory, George B.; Johnson, Alexander L.; et al.
Journal of Medicinal Chemistry, 1990 , vol. 33, # 5 p. 1312 - 1329