1: With acetic acid in benzene
T=100°C; Conrad-Limpach reaction;
2: in diphenylether; benzene
Conrad-Limpach reaction; 0.25 h; Reflux;
参考文献
Cross, R. Matthew; Monastyrskyi, Andrii; Mutka, Tina S.; Burrows, Jeremy N.; Kyle, Dennis E.; Manetsch, Roman
Journal of Medicinal Chemistry, 2010 , vol. 53, # 19 p. 7076 - 7094