N-苯甲酰基-D-苯丙氨酸合成路线 （共 30 条）
反应条件
1: Et3N / 0.17 h / 20 °C 2: CF3CO2H / 0.5 h View Scheme
参考文献
Ben-Ishai; Berger
Journal of Organic Chemistry, 1952 , vol. 17, p. 1564,1565
反应条件
1: 85 percent / LDA / tetrahydrofuran / -78 °C 2: 87 percent / 1N NaOH / methanol / 5 h / 60 °C View Scheme
参考文献
Schulthess, Adrian Heinz; Hansen, Hans-Juergen
Helvetica Chimica Acta, 1981 , vol. 64, # 5 p. 1322 - 1336
反应条件
1: 58 percent / pyridine / 1 h / 90 °C 2: 3 percent KOH / ethanol / 1 h / Heating View Scheme
参考文献
Noguchi; Mochida; Shingu; et al.
Chemical and Pharmaceutical Bulletin, 1984 , vol. 32, # 9 p. 3584 - 3587
反应条件
1: 10 percent NaOH / 4 h 2: 58 percent / pyridine / 1 h / 90 °C 3: 3 percent KOH / ethanol / 1 h / Heating View Scheme
参考文献
Noguchi; Mochida; Shingu; et al.
Chemical and Pharmaceutical Bulletin, 1984 , vol. 32, # 9 p. 3584 - 3587
反应条件
potassium hydroxide in ethanol 1 h; Heating;
参考文献
Noguchi; Mochida; Shingu; et al.
Chemical and Pharmaceutical Bulletin, 1984 , vol. 32, # 9 p. 3584 - 3587
反应条件
1: 97 percent / 1-ethyl-3-(3'-dimethylaminopropyl)carbodiimide hydrochloride / dimethylformamide / 0.17 h / 20 °C 2: 97 percent / K2CO3 / CH2Cl2; H2O / 2 h / 20 °C View Scheme
参考文献
Fujisaki, Fumiko; Oishi, Marumi; Sumoto, Kunihiro
Chemical and Pharmaceutical Bulletin, 2007 , vol. 55, # 1 p. 124 - 127
反应条件
water; oxonium T=25°C; different reaction conditions; solvent effect; Rate constantProduct distribution;
参考文献
Daffe, Viviane; Fastrez, Jacques
Journal of the Chemical Society, Perkin Transactions 2: Physical Organic Chemistry (1972-1999), 1983 , p. 783 - 788
反应条件
sodium hydroxide 0.5 h; Heating;
参考文献
Sikdar, Atul P.; Chetri, Ajoy B.; Das, Pranab J.
Indian Journal of Chemistry - Section B Organic and Medicinal Chemistry, 2003 , vol. 42, # 11 p. 2878 - 2881
反应条件
T=20°C; Hydrogenation;
参考文献
Waser
Helvetica Chimica Acta, 1925 , vol. 8, p. 124
参考文献
Ruggli; Ratti; Henzi
Helvetica Chimica Acta, 1929 , vol. 12, p. 351
