1: With Na2CO3*H2O; sodium carbonate T=35°C; 2: With chlorine T=35 - 40°C; 3 h; 3: With hydrogenchloride in water SolventReagent/catalyst;
参考文献
Bridge, Andrew W.; Jones, Ronald H.; Kabir, Humayun; Kee, Alex A.; Lythgoe, David J.; Nakach, Mustafa; Pemberton, Clive; Wrightman, John A.
Organic Process Research and Development, 2001 , vol. 5, # 1 p. 9 - 15
N-ethyl-N,N-diisopropylamine in acetonitrile 20 h; Heating;
参考文献
Saari, Walfred S.; Wai, John S.; Fisher, Thorsten E.; Thomas, Craig M.; Hoffman, Jacob M.; et al.
Journal of Medicinal Chemistry, 1992 , vol. 35, # 21 p. 3792 - 3802