2-氯-苯并噻唑-4-羰酰氯合成路线 (共 2 条)
参考文献
SIRTRIS PHARMACEUTICALS, INC.; VU, Chi, B.
Patent: WO2010/19606 A1, 2010 ;
Location in patent: Page/Page column 85-86 ;
WO 2010/019606 A1
反应条件
phosphorus pentachloride; trichlorophosphate in N,N-dimethyl-formamide
3 h; Reflux;
参考文献
SIRTRIS PHARMACEUTICALS, INC.; VU, Chi, B.
Patent: WO2010/19606 A1, 2010 ;
Location in patent: Page/Page column 85-86 ;
WO 2010/019606 A1