反应条件
1: 2,4,6-trichloro-pyrimidine With copper(l) iodide in tetrahydrofuran
Inert atmosphere;
2: ethylmagnesium bromide in tetrahydrofuran
T=0 - 20°C; 14 h;
参考文献
Boehringer Ingelheim International GmbH; EICKMEIER, Christian; GERLACH, Kai; HEINE, Niklas; WEBER, Alexander; GROSS, Ulrike
Patent: US2013/225593 A1, 2013 ;
Location in patent: Paragraph 0394-0396 ;