2-氯甲基-1,3-苯并噻唑合成路线 （共 34 条）
反应条件
triphenylphosphine in tetrachloromethane; benzene 2 h; Heating;
参考文献
Dondoni, Alessandro; Fantin, Giancarlo; Fogagnolo, Marco; Medici, Alessandro; Pedrini, Paola
Tetrahedron, 1988 , vol. 44, # 7 p. 2021 - 2032
反应条件
in toluene T=20°C; 16 h;
参考文献
Peprah, Kwakye; Zhu, Xue Y.; Eyunni, Suresh V.K.; Etukala, Jagan R.; Setola, Vincent; Roth, Bryan L.; Ablordeppey, Seth Y.
Bioorganic and Medicinal Chemistry, 2012 , vol. 20, # 5 p. 1671 - 1678
反应条件
boron trifluoride diethyl etherate in dichloromethane T=20°C; Inert atmosphere;
参考文献
Bastug, Gulluzar; Eviolitte, Christophe; Marko, Istvan E.
Organic Letters, 2012 , vol. 14, # 13 p. 3502 - 3505
反应条件
in dichloromethane Ambient temperature;
参考文献
American Home Products Corporation
Patent: US4594425 A1, 1986 ;
参考文献
American Home Products Corporation
Patent: US4876346 A1, 1989 ;
反应条件
methanesulfonic acid; silica gel T=140°C; 2.5 h;
参考文献
Sharghi, Hashem; Asemani, Omid
Synthetic Communications, 2009 , vol. 39, # 5 p. 860 - 867
反应条件
in dichloromethane T=0 - 20°C;
参考文献
Sheng, Chunquan; Che, Xiaoying; Wang, Wenya; Wang, Shengzheng; Cao, Yongbing; Yao, Jianzhong; Miao, Zhenyuan; Zhang, Wannian
European Journal of Medicinal Chemistry, 2011 , vol. 46, # 5 p. 1706 - 1712
反应条件
trichloroisocyanuric acid in chloroform Heating;
参考文献
Meltzer-Mats, Ella; Babai-Shani, Gali; Pasternak, Lily; Uritsky, Neta; Getter, Tamar; Viskind, Olga; Eckel, Juergen; Cerasi, Erol; Senderowitz, Hanoch; Sasson, Shlomo; Gruzman, Arie
Journal of Medicinal Chemistry, 2013 , vol. 56, # 13 p. 5335 - 5350
参考文献
PFIZER INC.
Patent: EP313202 A3, 1989 ;
反应条件
trichloroisocyanuric acid in dichloromethane 5 h; Heating;
参考文献
Ohba; Kosaka; Wakabayashi
Synthetic Communications, 1995 , vol. 25, # 21 p. 3421 - 3426
