1,2-苯并异噁唑-3-乙酸合成路线 (共 2 条)
反应条件
T=130°C; 0.5 h; Product distribution / selectivity;
参考文献
Sequoia Pharmaceuticals
Patent: US2005/267074 A1, 2005 ;
Location in patent: Page/Page column 26; 45 ;
反应条件
bromine in acetic acid
参考文献
Gianella,M. et al.
Chimica Therapeutica, 1972 , p. 127 - 132