反应条件
1: 2,4(3H,5H)-Thiazoledione With lithium diisopropyl amide in tetrahydrofuran; n-heptane; benzene
T=-78°C; 0.416667 h;
2: methyl iodide in tetrahydrofuran; n-heptane; benzene
T=-78°C; 2 h;
参考文献
BRISTOL-MYERS SQUIBB COMPANY; JOHNSON, James A.; JIANG, Ji; KIM, Soong-Hoon; PI, Zulan; QIAO, Jennifer X.; TORA, George O.; WANG, Tammy C.; FINLAY, Heather
Patent: WO2014/11513 A1, 2014 ;
Location in patent: Paragraph 00192 ;