反应条件
1: 4-(3-hydroxypropyl)-1-methylpiperazine With sodium hydride in N,N-dimethyl-formamide T=100°C; 0.0833333 h; 2: 4-[(2,4-dichloro-5-methoxyphenyl)amino]-7-fluoro-6-methoxy-3-quinolinecarbonitrile in N,N-dimethyl-formamide T=120°C; 2 h;
参考文献
Boschelli, Diane H.; Wang, Yanong D.; Johnson, Steve; Wu, Biqi; Ye, Fei; Barrios Sosa, Ana Carolina; Golas, Jennifer M.; Boschelli, Frank
Journal of Medicinal Chemistry, 2004 , vol. 47, # 7 p. 1599 - 1601