2,3-二氢-1H-茚-1-乙酸合成路线 （共 18 条）
反应条件
1: KOH / ethanol / Heating
2: polyphosphoric acid / Heating
3: zinc amalgam, aq. HCl / benzene / Heating
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参考文献
Pramanik; Mukherjee
Journal of the Indian Chemical Society, 1997 , vol. 74, # 9 p. 734 - 735
反应条件
1: piperidine / 72 h / 30 - 40 °C
2: KOH / ethanol / Heating
3: polyphosphoric acid / Heating
4: zinc amalgam, aq. HCl / benzene / Heating
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参考文献
Pramanik; Mukherjee
Journal of the Indian Chemical Society, 1997 , vol. 74, # 9 p. 734 - 735
反应条件
1: 75 percent / diethyl ether / 1.75 h
2: 69 percent / CF3CO3H, Na2HPO4 / CH2Cl2 / 4 h / Heating
3: 90 percent / 25percent aq. NaOH / 4 h / Heating
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参考文献
Lorentzen, Ronald J.; Brewster, James H.; Smith, Howard E.
Journal of the American Chemical Society, 1992 , vol. 114, # 6 p. 2181 - 2187
反应条件
1: 98 percent / SOCl2, NH3
2: 88 percent / P2O5 / Heating
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参考文献
Data; Taylor; Forcione
Journal of Pharmaceutical Sciences, 1974 , vol. 63, # 6 p. 848 - 853
反应条件
1: LiAlH4
2: HBr
3: (i) NaOEt, (ii) /BRN= 2440395/
4: (i) aq. KOH, (ii) aq. HCl
5: polyphosphoric acid
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参考文献
Anderson,A.G. et al.
Journal of Organic Chemistry, 1973 , vol. 38, # 8 p. 1439 - 1444
反应条件
1: 98 percent / SOCl2, NH3
2: 88 percent / P2O5 / Heating
3: 65 percent / NaN3, NH4Cl / dimethylformamide / 120 - 150 °C
View Scheme
参考文献
Roy, A.; Gupta, J. K.; Lahiri, S.C.
Journal of the Indian Chemical Society, 1983 , vol. 60, p. 377 - 380
反应条件
thionyl chloride; ammonia
参考文献
Roy, A.; Gupta, J. K.; Lahiri, S.C.
Journal of the Indian Chemical Society, 1983 , vol. 60, p. 377 - 380
反应条件
lithium aluminium tetrahydride
参考文献
Anderson,A.G. et al.
Journal of Organic Chemistry, 1973 , vol. 38, # 8 p. 1439 - 1444
