N-环丙基-N-(哌啶-4-基)-3-(三氟甲基)苯磺胺合成路线 (共 2 条)
反应条件
ammonium formate; palladium 10 on activated carbon in ethanol; water
2 h; Heating / reflux;
参考文献
EURO-CELTIQUE S.A.
Patent: WO2007/118853 A1, 2007 ;
Location in patent: Page/Page column 155-156 ;
WO 2007/118853 A1
反应条件
triethylamine in dichloromethane
T=0 - 20°C; 16 h; Product distribution / selectivity;
参考文献
EURO-CELTIQUE S.A.
Patent: WO2007/118853 A1, 2007 ;
Location in patent: Page/Page column 159-160 ;
WO 2007/118853 A1