反应条件
1: 85 percent / Ti(OiPr)4, 2-OH-3,5-Cl2-C6H4-CH=(t-Leu-Thr(OtBu)-Gly-OMe), iPrOH / toluene / 20 h / 4 °C 2: 6N HCl / 12 h / 70 °C View Scheme
参考文献
Krueger, Clinton A.; Kuntz, Kevin W.; Dzierba, Carolyn D.; Wirschun, Wolfgang G.; Gleason, John D.; Snapper, Marc L.; Hoveyda, Amir H.
Journal of the American Chemical Society, 1999 , vol. 121, # 17 p. 4284 - 4285