反应条件
1.1: 81 percent / triethyl(methoxycarbonylsulfamoyl)ammonium hydroxide / tetrahydrofuran / 0.25 h / 25 °C 2.1: LDA; NMPA / tetrahydrofuran; hexane 2.2: fluoromethoxyborane diethyl etherate; H2O2 (30percent); NaOH (3.0 M) / tetrahydrofuran / 2 h / 25 °C 2.3: 41 percent / pyridine / CH2Cl2 / 3 h / 25 °C View Scheme
参考文献
Rauchschwalbe, Guenter; Zellner, Armin; Schlosser, Manfred
European Journal of Organic Chemistry, 2001 , # 20 p. 3903 - 3909