1: 60 percent / 90 °C
2: 85 percent / iodine / CHCl3 / 25 °C
View Scheme
参考文献
Vasselin, David A.; Westwell, Andrew D.; Matthews, Charles S.; Bradshaw, Tracey D.; Stevens, Malcolm F. G.
Journal of Medicinal Chemistry, 2006 , vol. 49, # 13 p. 3973 - 3981