1: With triethylamine in dichloromethane T=0 - 20°C; 24 h; 2: With pyridine; 1,8-diazabicyclo[5.4.0]undec-7-ene in tetrachloromethane; acetonitrile 3 h; 3: With lithium aluminium tetrahydride
参考文献
ZAPAQ, INC.; THE BOARD OF TRUSTEES OF THE UNIVERSITY OF ILLINOIS; OKLAHOMA MEDICAL RESEARCH FOUNDATION
Patent: WO2006/34277 A1, 2006 ;
Location in patent: Page/Page column 61 ;
WO 2006/034277 A1