吲哚-4-羧酸甲酯合成路线

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Somei; Inoue; Tokutake; et al.
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123191-00-41-(三异丙基硅基)吲哚+

79-22-1氯甲酸甲酯

39830-66-5吲哚-4-羧酸甲酯

参考文献

Beswick; Greenwood; Mowlem; Nechvatal; Widdowson
Tetrahedron, 1988 , vol. 44, # 23 p. 7325 - 7334

39830-66-5吲哚-4-羧酸甲酯

49839-99-84-(2-硝基乙烯基)吲哚

参考文献

Maryanoff, Bruce E.; McComsey, David F.; Martin, Gregory E.; Shank, Richard P.
Bioorganic and Medicinal Chemistry Letters, 1998 , vol. 8, # 8 p. 983 - 988

39830-66-5吲哚-4-羧酸甲酯

433728-79-13-甲酸基-4-吲唑羧酸甲酯

参考文献

US2009/298809 A1, ;

Page/Page column 17-18 ;
US 20090298809 A1

39830-66-5吲哚-4-羧酸甲酯

90924-46-22-氧化吲哚-4-甲酸甲酯

参考文献

Taylor, Steven J.; Padyana, Anil K.; Abeywardane, Asitha; Liang, Shuang; Hao, Ming-Hong; De Lombaert, Stephane; Proudfoot, John; Farmer, Bennett S.; Li, Xiang; Collins, Brandon; Martin, Leslie; Albaugh, Daniel R.; Hill-Drzewi, Melissa; Pullen, Steven S.; Takahashi, Hidenori
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39830-66-5吲哚-4-羧酸甲酯

90924-06-41-甲基-1H-吲哚-4-羧酸

参考文献

Rigby, James H.; Burke, Patrick J.
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39830-66-5吲哚-4-羧酸甲酯

220499-12-7N-boc-4-羟基甲基吲哚

参考文献

NOVARTIS AG; BERST, Frederic; FURET, Pascal; MARZINZIK, Andreas; STAUFFER, Frederic
Patent: WO2011/157793 A1, 2011 ;
WO 2011/157793 A1

39830-66-5吲哚-4-羧酸甲酯+

24424-99-5二碳酸二叔丁酯

220499-11-61-BOC-吲哚-4-羧酸甲酯

参考文献

NOVARTIS AG; BERST, Frederic; FURET, Pascal; MARZINZIK, Andreas; STAUFFER, Frederic
Patent: WO2011/157793 A1, 2011 ;
Location in patent: Page/Page column 46-47 ;
WO 2011/157793 A1

39830-66-5吲哚-4-羧酸甲酯

220499-13-84-溴甲基-1H-吲哚-1-羧酸-1,1-二甲基乙酯

参考文献

NOVARTIS AG; BERST, Frederic; FURET, Pascal; MARZINZIK, Andreas; STAUFFER, Frederic
Patent: WO2011/157793 A1, 2011 ;
WO 2011/157793 A1

39830-66-5吲哚-4-羧酸甲酯+

68-12-2N,N-二甲基甲酰胺

53462-88-73-醛基-1H-吲哚-4-甲酸甲酯

参考文献

LABORATORIOS DEL DR. ESTEVE, S.A.; DRACONIS PHARMA, S.L.; ALMIRALL, S.A.; TORRENS JOVER, Andoni; MERCÈ VIDAL, Ramon; CALDENTEY FRONTERA, Francesc Xavier; RODRÍGUEZ GARRIDO, Antonio, David; CARCELLER GONZÁLEZ, Elena; SALAS SOLANA, Jordi
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Location in patent: Page/Page column 82 ;