反应条件
1: 92 percent
2: 80 percent / potassium tert-butoxide / 1.) 0.25 h, 2.) heating, 4 h
3: 40 percent / 1.) potassium carbonate / acetone / Heating; 1.) 0.5 h, 2.) 24 h
View Scheme
参考文献
Sherlock, Margaret H.; Kaminski, James J.; Tom, Wing C.; Lee, Joe F.; Wong, Shing-Chun; et al.
Journal of Medicinal Chemistry, 1988 , vol. 31, # 11 p. 2108 - 2121