反应条件
ammonia; 1,1'-carbonyldiimidazole
1.) CH2Cl2, reflux, 30 min, 2.) CH2Cl2, RT, 18 h; Multistep reaction;
参考文献
Jacobs, Robert T.; Bernstein, Peter R.; Cronk, Laura A.; Vacek, Edward P.; Newcomb, Lisa F.; et al.
Journal of Medicinal Chemistry, 1994 , vol. 37, # 9 p. 1282 - 1297