反应条件
1: 88 percent / NH3/EtOH / 1.5 h 2: 84 percent / NaN3 / dimethylformamide / 45 h / 80 °C 3: 66 percent / NH3, MeOH / 40 h / Ambient temperature 4: 70 percent / H2 / Pd-C / ethanol / 5 h / 2327.2 Torr View Scheme
参考文献
Ceulemans; Vandendriessche; Rozenski; Herdewijn
Nucleosides and Nucleotides, 1995 , vol. 14, # 1-2 p. 117 - 127