环丙基硼酸合成路线

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MSD Oss B.V.; Man, de, Adrianus, Petrus, Antonius; Sterrenburg, Jan-Gerard; Raaijmakers, Hans C.A.; Kaptein, Allard; Oubrie, Arthur A.; Rewinkel, Johannes, Bernardus, Maria; Jans, Christiaan, Gerardus, Johannes, Maria; Wijkmans, Jacobus C.H.M.; Barf, Tjeerd A.; Gao, Xiaolei; Boga, Sobhana Babu; Yao, Xin; Zhu, Hugh Y.; Cooper, Allen B.; Kim, Ronald M.
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19798-80-22-氨基-4-氯吡啶+

411235-57-9环丙基硼酸

908269-97-64-环丙基吡啶-2-胺

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MERCK SHARP and DOHME CORP.; MERCK CANADA INC.; DESCHENES, Denis; ALTMAN, Michael, D.; ELLIS, John Michael; FISCHER, Christian; HAIDLE, Andrew, M.; KATTAR, Solomon, D.; NORTHRUP, Alan, B.; SCHELL, Adam, J.; SMITH, Graham, F.; TAOKA, Brandon, M.; BIENSTOCK, Corey; DI FRANCESCO, Maria Emilia; DONOFRIO, Anthony; PETERSON, Scott; SPENCER, Kerrie, B.; JEWELL, James Patrick; ALI, Amjad; BENNETT, David Jonathan; DANG, Qun; WAI, John
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WO 2012/154518 A1

917899-39-9N,N-二甲基-5-碘-1H-吡唑-1-磺酰胺+

411235-57-9环丙基硼酸

917899-40-2

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ASTEX THERAPEUTICS LIMITED; THE INSTITUTE OF CANCER RESEARCH: ROYAL CANCER HOSPITAL; CANCER RESEARCH TECHNOLOGY LIMITED; ASTRAZENECA AB
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WO 2006/136830 A1

6602-54-62-氯-3-氰基吡啶+

411235-57-9环丙基硼酸

921760-69-2

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MERCK and CO., INC.; BANYU PHARMACEUTICAL CO., LTD.
Patent: WO2007/11809 A1, 2007 ;
Location in patent: Page/Page column 98 ;

128071-75-02-溴-3-吡啶甲醛+

411235-57-9环丙基硼酸

921760-70-5

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ASTLES, Peter Charles; GUIDETTI, Rossella; TIDWELL, Michael Wade; HOLLINSHEAD, Sean Patrick
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Location in patent: Page/Page column 9 ;
US 20100160288 A1

921760-93-2+

411235-57-9环丙基硼酸

921760-94-3

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MERCK and CO., INC.; BANYU PHARMACEUTICAL CO., LTD.
Patent: WO2007/11809 A1, 2007 ;
Location in patent: Page/Page column 104 ;

106-38-7对溴甲苯+

411235-57-9环丙基硼酸

6921-43-3

参考文献

Lemhadri, Mhamed; Doucet, Henri; Santelli, Maurice
Synthetic Communications, 2006 , vol. 36, # 1 p. 121 - 128

943320-69-2+

411235-57-9环丙基硼酸

943320-68-1

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Huang, Wei-Sheng; Metcalf, Chester A.; Sundaramoorthi, Raji; Wang, Yihan; Zou, Dong; Thomas, R. Mathew; Zhu, Xiaotian; Cai, Lisi; Wen, David; Liu, Shuangying; Romero, Jan; Qi, Jiwei; Chen, Ingrid; Banda, Geetha; Lentini, Scott P.; Das, Sasmita; Xu, Qihong; Keats, Jeff; Wang, Frank; Wardwell, Scott; Ning, Yaoyu; Snodgrass, Joseph T.; Broudy, Marc I.; Russian, Karin; Zhou, Tianjun; Commodore, Lois; Narasimhan, Narayana I.; Mohemmad, Qurish K.; Iuliucci, John; Rivera, Victor M.; Dalgarno, David C.; Sawyer, Tomi K.; Clackson, Tim; Shakespeare, William C.
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13534-89-9+

411235-57-9环丙基硼酸

944718-27-8

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SCHERING CORPORATION
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Location in patent: Page/Page column 158 ;
WO 2007/084451 A1

3934-20-1+

411235-57-9环丙基硼酸

954237-31-1

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MERCK SHARP and DOHME CORP.; EDMONDSON, Scott, D.; CHANG, Lehua; KAR, Nam Fung; MORRIELLO, Gregori, J.; MOYES, Christopher, J.; SHEN, Dong-Ming; ZHU, Cheng; ANTHONY, Neville, J.; JONES, Philip; SMITH, Graham, F.; SCOTT, Mark, E.; THOMPSON, Christopher, F.; JUNG, Joon; CAMMARANO, Carolyn; HOFFMAN, Dawn Marie
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WO 2011/025774 A1