3-[(4-氯苄基)磺酰基]-1H-1,2,4-噻唑-5-胺合成路线 (共 2 条)
反应条件
hydrazine in methanol 10 h; Heating;
参考文献
Reiter, J.; Somorai, T.; Jerkovich, Gy.; Dvortsak, P.
Journal of Heterocyclic Chemistry, 1982 , vol. 19, p. 1157 - 1164
反应条件
sodium hydroxide in ethanol T=70 - 75°C; 0.333333 h;
参考文献
Novinson; Springer; O'Brien; Scholten; Miller; Robins
Journal of Medicinal Chemistry, 1982 , vol. 25, # 4 p. 420 - 426