5-苯基-1H-氮杂革-2(3H)-酮合成路线 (共 2 条)
反应条件
water in ethanol
T=150°C; 20 h; Heating / reflux; Product distribution / selectivity;
参考文献
ELI LILLY AND COMPANY
Patent: WO2009/23453 A1, 2009 ;
Location in patent: Page/Page column 8-9 ;
WO 2009/023453 A1
反应条件
water in V methoxymethyl ester
108 h; Heating / reflux; Product distribution / selectivity;
参考文献
ELI LILLY AND COMPANY
Patent: WO2009/23453 A1, 2009 ;
Location in patent: Page/Page column 7-8 ;
WO 2009/023453 A1