反应条件
1: 25 percent / K2CO3, KI / dimethylformamide / 3 h / 40 °C
2: SnCl2, 5 N aq. HCl / ethanol / 16 h / 50 °C
View Scheme
参考文献
Madsen, Peter; Knudsen, Lotte B.; Wiberg, Finn C.; Carr, Richard D.
Journal of Medicinal Chemistry, 1998 , vol. 41, # 26 p. 5150 - 5157