反应条件
1: caesium carbonate / N,N-dimethyl-formamide / 0.25 h / 130 °C 2: AlCl3, aluminium chloride / dichloromethane / 0.5 h / 0 °C View Scheme
参考文献
MERCK SHARP and DOHME CORP.; DUFFY, Joseph, L.; BAO, Jianming; ONDEYKA, Debra, L.; TYAGARAJAN, Sriram; SHAO, Patrick; YE, Feng; KATIPALLY, Revathi; FINKE, Paul, E.; ZANG, Yi; PLOTKIN, Michael, A.; ROMERO, F. Anthony; MONINGKA, Remond; HUSSAIN, Zahid
Patent: WO2011/146324 A1, 2011 ;
WO 2011/146324 A1