1: 4-chloro-aniline With hydrogenchloride in water; acetone 2: With sodium nitrite in water; acetone 0.0416667 h; Sonication; 3: ethyl vinyl ether Further stages;
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Chernyak, Natalia; Buchwald, Stephen L.
Journal of the American Chemical Society, 2012 , vol. 134, # 43 p. 18147 - 18147,1
Dess-Martin periodane in dichloromethane T=20°C; 2.25 h;
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Cinelli, Maris A.; Li, Huiying; Chreifi, Georges; Martasek, Pavel; Roman, Linda J.; Poulos, Thomas L.; Silverman, Richard B.
Journal of Medicinal Chemistry, 2014 , vol. 57, # 4 p. 1513 - 1530
iodosylbenzene; 1-butylpyridinium tetrafluoroborate; [MnIIIT(N-Me-4-Py)P][PF6]5 T=30°C; 4 h; in open air; Title compound not separated from byproducts.;
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Saha, Rajat; Joarder, Biplab; Roy, Anupam Singha; Manirul Islam, Sk.; Kumar, Sanjay
Chemistry - A European Journal, 2013 , vol. 19, # 49 p. 16607 - 16614