反应条件
1: With (1,1'-bis(diphenylphosphino)ferrocene)palladium(II) dichloride; potassium acetate; 5,5,5',5'-tetramethyl-[2,2']bi[[1,3,2]dioxaborinanyl] in 1,4-dioxane; dichloromethane
T=80°C; 24 h;
2: With hydrogenchloride
T=40°C; 0.5 h;
参考文献
Lewis, Richard T.; Blackaby, Wesley P.; Blackburn, Timothy; Jennings, Andrew S. R.; Pike, Andrew; Wilson, Rowan A.; Hallett, David J.; Cook, Susan M.; Ferris, Pushpinder; Marshall, George R.; Reynolds, David S.; Sheppard, Wayne F. A.; Smith, Alison J.; Sohal, Bindi; Stanley, Joanna; Tye, Spencer J.; Wafford, Keith A.; Atack, John R.
Journal of Medicinal Chemistry, 2006 , vol. 49, # 8 p. 2600 - 2610