2-氯-1-[4-(嘧啶-2-基)哌嗪-1-基]乙酮合成路线 (共 2 条)
反应条件
N-ethyl-N,N-diisopropylamine in 1,4-dioxane
T=20°C; 2.5 h; Reflux;
参考文献
Sharma, Mani; Gupta, Monica; Singh, Divya; Kumar, Manoj; Kaur, Punit
Chemical Biology and Drug Design, 2013 , vol. 82, # 2 p. 156 - 166
反应条件
in ethanol
18 h; Reflux;
参考文献
Gilead Sciences, Inc.
Patent: US2012/289493 A1, 2012 ;
Location in patent: Page/Page column 84 ;
US 20120289493 A1