1: 7-amino-8-nitroquinoline With sodium hydride in tetrahydrofuran; mineral oil T=20°C; 0.5 h; 2: methyl iodide in tetrahydrofuran; mineral oil T=20°C; 5 h;
参考文献
Sunovion Pharmaceuticals Inc.
Patent: US2012/178748 A1, 2012 ;
Location in patent: Page/Page column 42 ;
US 20120178748 A1