6-碘咪唑并[1,2-a]吡啶合成路线 （共 3 条）
反应条件
in water; acetonitrile 14 h; Heating / reflux;
参考文献
ELI LILLY AND COMPANY
Patent: WO2004/50659 A1, 2004 ;
Location in patent: Page 64 ;
WO 2004/050659 A1
反应条件
in ethanol 3 h; Heating;
参考文献
Enguehard, Cecile; Hervet, Maud; Thery, Isabelle; Renou, Jean-Louis; Fauvelle, Florence; Gueiffier, Alain
Helvetica Chimica Acta, 2001 , vol. 84, # 12 p. 3610 - 3615
反应条件
copper(l) iodide; 1,10-phenanthroline; caesium carbonate in toluene
T=120°C;
参考文献
Daiichi Sankyo Company, Limited; AOKI, Kazumasa; MATSUI, Satoshi; YOSHIKAWA, Kenji; SHIMIZU,Hiroki; SASAKI, Junko; NAKAJIMA, Katsuyoshi; KANNO, Osamu; OIZUMI, Kiyoshi
Patent: EP2565185 A1, 2013 ;
Location in patent: Paragraph 0184 ;
