2-甲基-1,3-二氧代异吲哚啉-5-羧酸合成路线 (共 2 条)
反应条件
1: in tetrahydrofuran; water
T=20°C; 15 h;
2: With hydrogenchloride in water
pH=1;
参考文献
Takeda Chemical Industries, Ltd.
Patent: EP1466625 A1, 2004 ;
Location in patent: Page 164-165 ;
反应条件
in water
T=20 - 140°C;
参考文献
BOEHRINGER INGELHEIM PHARMA GMBH and CO. KG
Patent: WO2004/26829 A2, 2004 ;
Location in patent: Page/Page column 76 ;
WO 2004/026829 A2