反应条件
1: 60 percent / AlCl3, HCl / CH2Cl2 / 0.5 h / 0 °C
2: 1.) p-TsNHNH2, HCl, 2.) NaOMe / 1.) THF, reflux, 30 min, 2.) irradiation, 22 h
View Scheme
参考文献
Truesdale, E.A.; Cram, Donald J.
Journal of Organic Chemistry, 1980 , vol. 45, # 20 p. 3974 - 3981