反应条件
1: 2-acetyl-2H-[1,2,4]triazine-3,5-dione With sodium hydride in N,N-dimethyl-formamide
T=20°C; 0.5 h;
2: methyl iodide in N,N-dimethyl-formamide
6 h;
参考文献
Prabhakaran, Jaya; Parsey, Ramin V.; Majo, Vattoly J.; Hsiung, Shu-Chi; Milak, Matthew S.; Tamir, Hadassah; Simpson, Norman R.; Van Heertum, Ronald L.; Mann, J. John; Dileep Kumar
Bioorganic and Medicinal Chemistry Letters, 2006 , vol. 16, # 8 p. 2101 - 2104